| RESEARCH
Our
laboratory has long been interested on the mechanisms by which neurotransmitters
modulate the excitability of neuronal and glial cells. Molecular
effectors for such modulation are for example potassium channels,
a large and diverse class of transmembrane proteins that mediate
the controlled flux of potassium ions. Currently we are working
with the G protein-gated inwardly rectifying potassium (GIRK) channels.
GIRK channels open upon activation of metabotropic receptors (e.g.opioids,
muscarinic, adrenergic receptors) that couple to the Gi or Go class
of G proteins. We are employing the heterologous expression of GIRK
channels and various metabotropic receptors to investigate how this
signaling takes place.
Another
major effort in our laboratory aims to elucidate the role of inwardly
rectifying potassium channels in glial cell function. Glial buffering
of the extracellular potassium concentration in retina has been
elegantly demonstrated using electrophysiological methods. Inwardly
rectifying potassium channels in these glial cells are spatially
localized to optimally perform this function. Research in our laboratory
has established the essential role of Kir4.1 channel in mouse retina
for the buffering of extracellular potassium concentration. More
recently we have been investigating the role of accessory proteins
for the modulation and subcellular localization of Kir4.1 channels
in Müller cells. We have identified a potential macromolecular
complex (Aquaporin-4, Kir4.1 and alpha syntrophin) that hold this
cluster together.

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